{"product_id":"optimization-in-drug-discovery-in-vitro-methods-9781627037419","title":"Optimization in Drug Discovery: In Vitro Methods","description":"\u003cp\u003e • Author(s): Gary W. Caldwell\u003cbr\u003e • Publisher: Springer\u003cbr\u003e • Publisher Imprint: Humana\u003cbr\u003e • BISAC: Pharmacology\u003c\/p\u003e\u003cp\u003e\u003c\/p\u003e\u003cp\u003e\u003cb\u003eFrom the Back Cover\u003c\/b\u003e\u003cbr\u003e\u003c\/p\u003e\u003cp\u003eThoroughly revised and updated, \u003ci\u003eOptimization in Drug Discovery: In Vitro Methods, Second Edition\u003c\/i\u003e presents a wide spectrum of in vitro assays including formulation, plasma binding, absorption and permeability, cytochrome P450 (CYP) and UDP-glucuronosyltransferases (UGT) metabolism, CYP inhibition and induction, drug transporters, drug-drug interactions via assessment of reactive metabolites, genotoxicity, and chemical and photo-mutagenicity assays. Written for the \u003ci\u003eMethods in Pharmacology and Toxicology\u003c\/i\u003e series, chapters include introductions to their respective topics, lists of the necessary materials and reagents, step-by-step, readily reproducible protocols, and tips on troubleshooting and avoiding known pitfalls. Expert authors have developed and utilized these in vitro assays to achieve \"drug-like\" characteristics in addition to efficacy properties and good safety profiles of drug candidates. \u003c\/p\u003e\u003cp\u003e \u003c\/p\u003eComprehensive and up-to-date, \u003ci\u003eOptimization in Drug Discovery: In Vitro Methods, Second Edition\u003c\/i\u003e aims to guide researchers down the difficult path to successful drug discovery and development.","brand":"Springer","offers":[{"title":"Hardcover","offer_id":45277280895127,"sku":"9781627037419","price":14553.0,"currency_code":"INR","in_stock":true}],"thumbnail_url":"\/\/cdn.shopify.com\/s\/files\/1\/0666\/3471\/1191\/files\/9781627037419.webp?v=1769288024","url":"https:\/\/atlanticbooks.com\/products\/optimization-in-drug-discovery-in-vitro-methods-9781627037419","provider":"Atlantic Books","version":"1.0","type":"link"}